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Home > Encyclopedia > 6-Benzothiazoleaceticacid,2-amino-(8CI,9CI)

6-Benzothiazoleaceticacid,2-amino-(8CI,9CI)

6-Benzothiazoleaceticacid,2-amino-(8CI,9CI) structure

6-Benzothiazoleaceticacid,2-amino-(8CI,9CI) 

structure
  • CAS No:

    30132-15-1

  • Formula:

    C9H8N2O2S

  • Chemical Name:

    6-Benzothiazoleaceticacid,2-amino-(8CI,9CI)

  • Synonyms:

    (2-Aminobenzothiazol-6-yl)acetic acid;2-(2-Aminobenzo[d]thiazol-6-yl)acetic acid;(2-Amino-benzothiazol-6-yl)-acetic acid;2-aminobenzothiazole-6-acetic acid;2-(2-amino-1,3-benzothiazol-6-yl)acetic acid;6-Benzothiazoleacetic acid, 2-amino-;(2-amino-1,3-benzothiazol-6-yl)acetic acid;2-Amino-6-(carboxymethyl)benzothiazole;2-(2-aminobenzothiazol-6-yl)acetic acid;TimTec1_007304

  • Categories:

    Pharmaceutical Intermediates  >  Heterocyclic Compound

6-Benzothiazoleaceticacid,2-amino-(8CI,9CI) Basic Attributes

208.23702

208.031

Characteristics

104

1.5

1.531±0.06 g/cm3

263 - 264 °C

H2O: Very slightly soluble (0.6 g/L) (25 ºC)

6-Benzothiazoleaceticacid,2-amino-(8CI,9CI) Use and Manufacturing

A. A. To prepare the intermediate A solution of (2-ami'o-benzothiazol-6-yl)-acetic acid (0.61 mmol, as prepared by Meyer et al. in J. Med. Chem. 1997, 40, 1060) in absolute etha'ol (10 mL) was treated with 3 drops of concentrated H2SO4 and. ca. 1 g of dry 4 A molecular sieves, and EXAMPLE 8; 3-(2-Fluorophenyl)-4-(2-(isopropylamino)benzo[d]thiazol-6-yl)-lH-pyrazol-5-oI; 1. Methyl 2-(2-aminobenzo[d]thiazol-6-yl)acetate[00175] A mixture of B. To prepare the intermediate methyl (2-amino-benzothiazol-6-yl)acetate, 2 mL concentrated H2SO4 was added dropwise to a solution of

Computed Properties

Molecular Weight:208.24
XLogP3:1.5
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:5
Rotatable Bond Count:2
Exact Mass:208.03064868
Monoisotopic Mass:208.03064868
Topological Polar Surface Area:104
Heavy Atom Count:14
Complexity:237
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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